(1R,3R)-N<sup>1</sup>-[5-(1-Ethylpropyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,3-cyclopentanediamine
Advanced Breast Cancer
Nuvation Bio Inc.Small moleculePhase 1/2Active
D
31/ 100
Provisional rating · Methodology v0.2
Rating breakdown
- Clinical Evidence
- 17/ 100
- Competitive Position
- 73/ 100
Competitive context
890 Active assets in the Advanced Breast Cancer cohort.
| Asset / Sponsor | Phase | Rating |
|---|---|---|
Lapatinib University of New Mexico | Phase 3 | BBB |
Darolutamide Vandana Abramson | Phase 2 | BBB |
Trastuzumab Duocarmazine Byondis B.V. | Phase 3 | BB |
ERIBULIN MONOMETHANESULFONATE Henan Cancer Hospital | Phase 4 | BB |
Palbociclib Hoffmann-La Roche | Phase 4 | BB |
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Same molecule, other indications
(1R,3R)-N<sup>1</sup>-[5-(1-Ethylpropyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,3-cyclopentanediamine is also rated in:
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